526522 | PIM1 Kinase Inhibitor IV

526522
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      Overview

      Replacement Information

      Key Spec Table

      Empirical FormulaCAS #
      C₁₇H₁₁ClN₄O477845-12-8

      Pricing & Availability

      Catalogue NumberAvailability Packaging Qty/Pack Price Quantity
      526522-5MG
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      In Stock 
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          Plastic ampoule 5 mg
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          Description
          OverviewA pyrimidinyl-benzisoxazolo compound that interacts with Lys67 and Glu121 at the PIM1 active site and inhibits PIM1 kinase activity with a Ki value of 0.091 µM.
          Catalogue Number526522
          Brand Family Calbiochem®
          Synonyms4-(3-(4-Chlorophenyl)-2,1-benzisoxazol-5-yl)-2-pyrimidinamine
          References
          ReferencesPierce, A.C., et al. 2008. J. Med. Chem. 51, 1972.
          Product Information
          CAS number477845-12-8
          FormYellow solid
          Hill FormulaC₁₇H₁₁ClN₄O
          Chemical formulaC₁₇H₁₁ClN₄O
          Structure formula ImageStructure formula Image
          Applications
          Biological Information
          Purity≥97% by HPLC
          Physicochemical Information
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          S PhraseS: 22-24/25

          Do not breathe dust.
          Avoid contact with skin and eyes.
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Ambient Temperature Only
          Toxicity Standard Handling
          Storage +2°C to +8°C
          Protect from Light Protect from light
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Packaging Information
          Packaged under inert gas Packaged under inert gas
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          SDS

          Title

          Safety Data Sheet (SDS) 

          Certificates of Analysis

          TitleLot Number
          526522

          References

          Reference overview
          Pierce, A.C., et al. 2008. J. Med. Chem. 51, 1972.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision18-April-2011 RFH
          Synonyms4-(3-(4-Chlorophenyl)-2,1-benzisoxazol-5-yl)-2-pyrimidinamine
          DescriptionA pyrimidinyl-benzisoxazolo compound that interacts with Lys67 and Glu121 at the PIM1 active site and inhibits PIM1 kinase activity with a Ki value of 0.091 µM.
          FormYellow solid
          Intert gas (Yes/No) Packaged under inert gas
          CAS number477845-12-8
          Chemical formulaC₁₇H₁₁ClN₄O
          Structure formulaStructure formula
          Purity≥97% by HPLC
          SolubilityDMSO (5 mg/ml)
          Storage +2°C to +8°C
          Protect from light
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Toxicity Standard Handling
          ReferencesPierce, A.C., et al. 2008. J. Med. Chem. 51, 1972.