05-22-3838 BQ-788, Sodium Salt - CAS - Calbiochem

05-22-3838
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      Overview

      Replacement Information

      Key Spec Table

      Empirical Formula
      C₃₄H₅₀N₅O₇Na

      Pricing & Availability

      Catalogue NumberAvailability Packaging Qty/Pack Price Quantity
      05-22-3838-1MG
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          Plastic ampoule 1 mg
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          05-22-3838-5MG
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              Plastic ampoule 5 mg
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              Description
              OverviewHighly selective ETB-receptor antagonist (IC50 = 1.2 nM).
              Catalogue Number05-22-3838
              Brand Family Calbiochem®
              SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
              References
              ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
              Taniai, H., et al. 2001. Hepatology 33, 894.
              Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
              Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
              Product Information
              ATP CompetitiveN
              FormWhite to off-white lyophilized solid
              Hill FormulaC₃₄H₅₀N₅O₇Na
              Chemical formulaC₃₄H₅₀N₅O₇Na
              ReversibleN
              Structure formula ImageStructure formula Image
              Applications
              Biological Information
              Primary TargetETB-receptor antagonist
              Primary Target IC<sub>50</sub>1.2 nM as ETB-receptor antagonist
              Purity≥95% by HPLC
              Physicochemical Information
              Cell permeableN
              Dimensions
              Materials Information
              Toxicological Information
              Safety Information according to GHS
              Safety Information
              Product Usage Statements
              Storage and Shipping Information
              Ship Code Ambient Temperature Only
              Toxicity Standard Handling
              Storage -20°C
              Protect from Moisture Protect from moisture
              Do not freeze Ok to freeze
              Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
              Packaging Information
              Transport Information
              Supplemental Information
              Specifications

              Documentation

              MSDS

              Title

              Safety Data Sheet (SDS) 

              Certificates of Analysis

              TitleLot Number
              05-22-3838

              References

              Reference overview
              Okada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
              Taniai, H., et al. 2001. Hepatology 33, 894.
              Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
              Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
              Data Sheet

              Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

              Revision18-September-2008 RFH
              SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
              DescriptionA highly selective and competitive ETB receptor antagonist (IC50 = 1.2 nM).
              FormWhite to off-white lyophilized solid
              Chemical formulaC₃₄H₅₀N₅O₇Na
              Structure formulaStructure formula
              Purity≥95% by HPLC
              SolubilityDMSO (2 mg/ml), Methanol:H₂O (3:1) (2 mg/ml), or 0.01% NH₄OH (1 mg/ml)
              Storage -20°C
              Protect from moisture
              Do Not Freeze Ok to freeze
              Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
              Toxicity Standard Handling
              ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
              Taniai, H., et al. 2001. Hepatology 33, 894.
              Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
              Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.