344150
FPT Inhibitor I
(E,E)-2-[(Dihydroxyphosphinyl)methyl]-3-oxo-3-[(3,7,11-trimethyl-2,6,10-dodecatrienyl)-amino]propanoic Acid, 3Na
Untuk pertanyaan umum, silakan hubungi Layanan Pelanggan kami:
Merck KGaA
Frankfurter Str. 250
64293 Darmstadt
Germany
Telefon: +49 6151 72-0
Faks: +49 6151 72 2000
31 May 2012
memuat
Potent and highly selective inhibitor of farnesyltransferase (FTase; IC50 = 83 nM). Inhibits geranylgeranyltransferase (GGTase) I and II at much higher concentrations (IC50 = 26 µM and 47 µM for GGTase I and II, respectively).
| Informasi produk | |||
|---|---|---|---|
| Form | White solid | ||
| Primary Target | FTase | ||
| Primary Target IC50 | 83 nM | ||
| Secondary target | geranylgeranyltransferase (GGTase) I and II at much higher concentrations (IC50 = 26 µM and 47 µM for GGTase I and II, respectively) | ||
| Hygrocopic | Ya | ||
| Packaged under inert gas | Ya | ||
| Purity | ≥85% by NMR | ||
| Formulasi kimia | C19H29NO6P · 3Na | ||
| Simpan dan kirim informasi | |||
|---|---|---|---|
| Penyimpanan | ≤ -70°C | ||
| Ship |
Ambient Temperature Only
Standard Handling |
||
