For general questions please contact our Customer Service:
Merck KGaA
Frankfurter Str. 250
64293 Darmstadt
Germany
Phone: +49 6151 72-0
Fax: +49 6151 72 2000
31 May 2012
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This product has been discontinued.
Please refer to our complete listing of protein phosphatase inhibitors for possible alternatives. Please read the alternative product documentation carefully and contact technical service if you need additional information.
A potent phosphotyrosine phosphatase inhibitor. Activates the insulin receptor kinase (IRK) in hepatoma cells. A potent competitive inhibitor of glucose-6-phosphatase (Ki = 420 nM in intact microsomes). Also reported to potently inhibit PTEN (IC50 = 31 nM).
| Product information | |||
|---|---|---|---|
| Form | Yellow solid | ||
| Primary Target | glucose-6-phophatase | ||
| Primary Target IC50 | 420 nM | ||
| Secondary target | PTEN (IC50 = 31 nM) | ||
| Molar mass | 367.3 | ||
| Protect from Light | Yes | ||
| Packaged under inert gas | Yes | ||
| Purity | ≥90% by 5¹V-NMR | ||
| Solubility | H2O | ||
| Chemical formula | K2[VO(O2)2C6H4NO2] · 2H2O | ||
| Store and ship information | |||
|---|---|---|---|
| Storage | -20°C | ||
| Ship |
Ambient Temperature Only
Standard Handling |
||
