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371780 GP Antagonist-2A - Calbiochem

371780
Purchase on Sigma-Aldrich

Overview

Replacement Information

Key Spec Table

Empirical Formula
C₇₉H₁₀₅N₂₁O₁₃S

Products

Catalogue NumberPackaging Qty/Pack
371780-1MG Plastic ampoule 1 mg
Description
OverviewA peptide that selectively inhibits the activation of Gq by M1-muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 µM. Blocks angiotensin II-stimulated sis-inducing factor and STAT3 tyrosine phosphorylation.
Catalogue Number371780
Brand Family Calbiochem®
SynonymsRPKPQQDWFDWDWM
References
ReferencesHunt, R.A., et al. 1999. Hypertension 34, 603.
Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.
Product Information
ATP CompetitiveN
FormLyophilized solid
FormulationSupplied as a trifluoroacetate salt.
Hill FormulaC₇₉H₁₀₅N₂₁O₁₃S
Chemical formulaC₇₉H₁₀₅N₂₁O₁₃S
ReversibleN
Quality LevelMQ100
Applications
Biological Information
Primary TargetInhibits the activation of Gq by M1-muscarinic cholinergic receptors
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Peptide SequenceH-Arg-Pro-Lys-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH₂
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications

Documentation

GP Antagonist-2A - Calbiochem SDS

Title

Safety Data Sheet (SDS) 

GP Antagonist-2A - Calbiochem Certificates of Analysis

TitleLot Number
371780

References

Reference overview
Hunt, R.A., et al. 1999. Hypertension 34, 603.
Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.
Data Sheet

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision13-May-2010 JSW
SynonymsRPKPQQDWFDWDWM
DescriptionA peptide that selectively inhibits the activation of Gq by M1-muscarinic cholinergic receptors. Also inhibits activation by cholecystokinin receptor in pancreatic acini at 10 µM. Blocks angiotensin II-stimulated sis-inducing factor and STAT3 tyrosine phosphorylation.
FormLyophilized solid
FormulationSupplied as a trifluoroacetate salt.
Chemical formulaC₇₉H₁₀₅N₂₁O₁₃S
Peptide SequenceH-Arg-Pro-Lys-Pro-Gln-Gln-D-Trp-Phe-D-Trp-D-Trp-Met-NH₂
Purity≥95% by HPLC
SolubilityH₂O (25 mg/ml)
Storage -20°C
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 1 month at -20°C.
Toxicity Standard Handling
ReferencesHunt, R.A., et al. 1999. Hypertension 34, 603.
Tsunoda Y., et al. 1995. Biochem. Biophys. Res. Commun. 211, 648.
Mukai, H., et al. 1992. J. Biol. Chem. 267, 16237.