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A highly selective and potent agonist for group II metabotropic glutamate receptor (EC50 = 0.4, 0.4, > 100, > 100, > 300 and > 300 µM for human mGlu2, mGlu3, mGlu1, mGlu5, mGlu4 and mGlu7 receptors respectively). Used as anti- and pro-convulsant, neuroprotectant, antinociceptive, and addiction treatment.
Folbergrová, J., et al. 2005. Experimental Neurology.192, 420. Fisher, K., et al. 2002. Pharmacol. Bioche. and Behav.73, 411. Schoepp, D., et al. 1995. Neuropharmacology.34, 843. Monn, J., et al. 1996. J. Med. Chem.39, 2990.
Product Information
CAS number
169209-63-6
Form
Off-white powder
Hill Formula
C₆H₁₀N₂O₄
Chemical formula
C₆H₁₀N₂O₄
Structure formula Image
Applications
Biological Information
Primary Target
mGlu₂ and mGlu₃
Purity
≥98% by HPLC
Physicochemical Information
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code
Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
Toxicity
Standard Handling
Storage
+2°C to +8°C
Protect from Light
Protect from light
Do not freeze
Ok to freeze
Special Instructions
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Folbergrová, J., et al. 2005. Experimental Neurology.192, 420. Fisher, K., et al. 2002. Pharmacol. Bioche. and Behav.73, 411. Schoepp, D., et al. 1995. Neuropharmacology.34, 843. Monn, J., et al. 1996. J. Med. Chem.39, 2990.
Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.
A highly selective and potent agonist for group II metabotropic glutamate receptor (EC50 = 0.4, 0.4, > 100, > 100, > 300 and > 300 µM for human mGlu2, mGlu3, mGlu1, mGlu5, mGlu4 and mGlu7 receptors respectively). Used as anti- and pro-convulsant, neuroprotectant, antinociceptive, and addiction treatment.
Form
Off-white powder
CAS number
169209-63-6
Chemical formula
C₆H₁₀N₂O₄
Structure formula
Purity
≥98% by HPLC
Solubility
H₂O (100 mM)
Storage
Protect from light
+2°C to +8°C
Do Not Freeze
Ok to freeze
Special Instructions
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Toxicity
Standard Handling
References
Folbergrová, J., et al. 2005. Experimental Neurology.192, 420. Fisher, K., et al. 2002. Pharmacol. Bioche. and Behav.73, 411. Schoepp, D., et al. 1995. Neuropharmacology.34, 843. Monn, J., et al. 1996. J. Med. Chem.39, 2990.
