5.05894
CGP 7930
Synonym(s):
CGP 7930, GABA B Receptor Antagonist, CGP7930, CGP 7930, CGP-7930
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About This Item
Empirical Formula (Hill Notation):
C19H32O2
CAS Number:
Molecular Weight:
292.46
MDL number:
UNSPSC Code:
12352200
NACRES:
NA.77
Assay:
≥98% (HPLC)
Form:
solid
Storage condition:
OK to freeze, protect from light
assay
≥98% (HPLC)
Quality Segment
form
solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze, protect from light
color
pale yellow
solubility
DMSO: 100 mM, ethanol: 100 mM
storage temp.
2-8°C
SMILES string
OCC(Cc1cc(c(c(c1)C(C)(C)C)O)C(C)(C)C)(C)C
InChI
1S/C19H32O2/c1-17(2,3)14-9-13(11-19(7,8)12-20)10-15(16(14)21)18(4,5)6/h9-10,20-21H,11-12H2,1-8H3
InChI key
XLWJPQQFJNGUPA-UHFFFAOYSA-N
General description
A blood brain barrier permeable, positive allosteric modulator of the metabotropic GABAB receptor. Shown to modulate GABAB receptor in the high affinity state and thereby increases agonist affinity for the receptor. Also enhances agonist potency and efficacy even on recombinant GABAB receptors. Exhibits anxiolytic effects in rodents.
Other Notes
Adams, C. et al., 2007. CNS Drug Rev.13, 308.
Pin, J.P., et al., 2007. Curr. Neuropharmacol.5, 195.
Pin, J.P., et al., 2007. Curr. Neuropharmacol.5, 195.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
Toxicity: Standard Handling (A)
Storage Class
11 - Combustible Solids
wgk
WGK 3
flash_point_f
Not applicable
flash_point_c
Not applicable
Certificates of Analysis (COA)
Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.
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