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05-22-3838 BQ-788, Sodium Salt - CAS - Calbiochem

05-22-3838
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Overview

Replacement Information

Key Spec Table

Empirical Formula
C₃₄H₅₀N₅O₇Na

Products

Catalogue NumberPackaging Qty/Pack
05-22-3838-1MG Plastic ampoule 1 mg
05-22-3838-5MG Plastic ampoule 5 mg
Description
OverviewHighly selective ETB-receptor antagonist (IC50 = 1.2 nM).
Catalogue Number05-22-3838
Brand Family Calbiochem®
SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
References
ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
Taniai, H., et al. 2001. Hepatology 33, 894.
Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
Product Information
ATP CompetitiveN
FormWhite to off-white lyophilized solid
Hill FormulaC₃₄H₅₀N₅O₇Na
Chemical formulaC₃₄H₅₀N₅O₇Na
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
Biological Information
Primary TargetETB-receptor antagonist
Primary Target IC<sub>50</sub>1.2 nM as ETB-receptor antagonist
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Standard Handling
Storage -20°C
Protect from Moisture Protect from moisture
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications

Documentation

BQ-788, Sodium Salt - CAS - Calbiochem SDS

Title

Safety Data Sheet (SDS) 

BQ-788, Sodium Salt - CAS - Calbiochem Certificates of Analysis

TitleLot Number
05-22-3838

References

Reference overview
Okada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
Taniai, H., et al. 2001. Hepatology 33, 894.
Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
Data Sheet

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision18-September-2008 RFH
SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
DescriptionA highly selective and competitive ETB receptor antagonist (IC50 = 1.2 nM).
FormWhite to off-white lyophilized solid
Chemical formulaC₃₄H₅₀N₅O₇Na
Structure formulaStructure formula
Purity≥95% by HPLC
SolubilityDMSO (2 mg/ml), Methanol:H₂O (3:1) (2 mg/ml), or 0.01% NH₄OH (1 mg/ml)
Storage -20°C
Protect from moisture
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
Toxicity Standard Handling
ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
Taniai, H., et al. 2001. Hepatology 33, 894.
Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.