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361555 GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem

361555
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Overview

Replacement Information

Key Spec Table

Empirical FormulaCAS #
C₁₈H₁₅N₅404828-08-6

Products

Catalogue NumberPackaging Qty/Pack
361555-1MG Plastic ampoule 1 mg
361555-5MG Plastic ampoule 5 mg
Description
OverviewAn aminopyrazole compound that acts as a potent and ATP-binding site inhibitor of GSK-3 with a Ki of 24 nM.
Catalogue Number361555
Brand Family Calbiochem®
Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
References
ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.
Product Information
CAS number404828-08-6
ATP CompetitiveN
FormWhite solid
Hill FormulaC₁₈H₁₅N₅
Chemical formulaC₁₈H₁₅N₅
ReversibleN
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
Biological Information
Primary TargetGSK-3
Primary Target K<sub>i</sub>24 nM against GSK-3
Purity≥95% by HPLC
Physicochemical Information
Cell permeableN
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Ambient Temperature Only
Toxicity Carcinogenic / Teratogenic
Storage +2°C to +8°C
Protect from Light Protect from light
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications

Documentation

GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem SDS

Title

Safety Data Sheet (SDS) 

GSK-3 Inhibitor XIII - CAS 404828-08-6 - Calbiochem Certificates of Analysis

TitleLot Number
361555

References

Reference overview
Pierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.
Data Sheet

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision01-July-2008 RFH
Synonyms(5-Methyl-1H-pyrazol-3-yl)-(2-phenylquinazolin-4-yl)amine
DescriptionA potent and ATP-competitive inhibitor of GSK-3 (Ki = 24 nM).
FormWhite solid
CAS number404828-08-6
Chemical formulaC₁₈H₁₅N₅
Structure formulaStructure formula
Purity≥95% by HPLC
SolubilityDMSO (5 mg/ml)
Storage +2°C to +8°C
Protect from light
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.
Toxicity Carcinogenic / Teratogenic
ReferencesPierce, A.C., et al. 2005. J. Med. Chem. 48, 1278.