05-22-3838 BQ-788, Sodium Salt - CAS - Calbiochem

05-22-3838
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Overview

Replacement Information

Key Spec Table

Empirical Formula
C₃₄H₅₀N₅O₇Na

Pricing & Availability

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05-22-3838-1MG
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      Plastic ampoule 1 mg
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      05-22-3838-5MG
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          Description
          OverviewHighly selective ETB-receptor antagonist (IC50 = 1.2 nM).
          Catalogue Number05-22-3838
          Brand Family Calbiochem®
          SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
          References
          ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
          Taniai, H., et al. 2001. Hepatology 33, 894.
          Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
          Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
          Product Information
          ATP CompetitiveN
          FormWhite to off-white lyophilized solid
          Hill FormulaC₃₄H₅₀N₅O₇Na
          Chemical formulaC₃₄H₅₀N₅O₇Na
          ReversibleN
          Structure formula ImageStructure formula Image
          Quality LevelMQ100
          Applications
          Biological Information
          Primary TargetETB-receptor antagonist
          Primary Target IC<sub>50</sub>1.2 nM as ETB-receptor antagonist
          Purity≥95% by HPLC
          Physicochemical Information
          Cell permeableN
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Ambient Temperature Only
          Toxicity Standard Handling
          Storage -20°C
          Protect from Moisture Protect from moisture
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          BQ-788, Sodium Salt - CAS - Calbiochem SDS

          Title

          Safety Data Sheet (SDS) 

          BQ-788, Sodium Salt - CAS - Calbiochem Certificates of Analysis

          TitleLot Number
          05-22-3838

          References

          Reference overview
          Okada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
          Taniai, H., et al. 2001. Hepatology 33, 894.
          Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
          Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision18-September-2008 RFH
          SynonymsN-cis-2,6-Dimethylpiperidinocarbonyl-L-γ-MeLeu-D-Trp(MeOCO)-D-Nle-OH, Na
          DescriptionA highly selective and competitive ETB receptor antagonist (IC50 = 1.2 nM).
          FormWhite to off-white lyophilized solid
          Chemical formulaC₃₄H₅₀N₅O₇Na
          Structure formulaStructure formula
          Purity≥95% by HPLC
          SolubilityDMSO (2 mg/ml), Methanol:H₂O (3:1) (2 mg/ml), or 0.01% NH₄OH (1 mg/ml)
          Storage -20°C
          Protect from moisture
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). DMSO and Methano:H₂O stock solutions are stable for up to 2 months at -20°C.
          Toxicity Standard Handling
          ReferencesOkada, M., and Nishikibe, M. 2002. Cardiovasc. Drug Reviews 20, 53.
          Taniai, H., et al. 2001. Hepatology 33, 894.
          Fukuroda, T., et al. 1994. Biochem. Biophys. Res. Commun. 199, 1461.
          Ishikawa, K., et al. 1994. Proc. Natl. Acad. Sci. USA 91, 4892.