217531 Sigma-AldrichCARM1 Inhibitor - CAS 1020399-49-8 - Calbiochem
The CARM1 Inhibitor controls the biological activity of CARM1. This small molecule/inhibitor is primarily used for Cell Structure applications.
More>> The CARM1 Inhibitor controls the biological activity of CARM1. This small molecule/inhibitor is primarily used for Cell Structure applications. Less<<Synonyms: PRMT Inhibitor V, Coactivator-Associated Arginine Methyltransferase 1 Inhibitor, 1-Benzyl-3,5-bis-(3-bromo-4-hydroxybenzylidene)piperidin-4-one, 3,5-bis(3-Bromo-4-hydroxybenzylidene)-1-benzylpiperidin-4-one
Recommended Products
Overview
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Key Spec Table
CAS # | Empirical Formula |
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1020399-49-8 | C₂₆H₂₁Br₂NO₃ |
Products
Catalogue Number | Packaging | Qty/Pack | |
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217531-10MG | Glass bottle | 10 mg |
References | |
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References | Cheng, D., et al. 2011. J. Med. Chem. 54, 4928. |
Product Information | |
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CAS number | 1020399-49-8 |
Form | Orange solid |
Hill Formula | C₂₆H₂₁Br₂NO₃ |
Chemical formula | C₂₆H₂₁Br₂NO₃ |
Reversible | Y |
Structure formula Image | |
Quality Level | MQ100 |
Applications |
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Biological Information | |
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Primary Target | PRMT4 |
Primary Target IC<sub>50</sub> | CARM1-mediated methylation over PRMT1 and SET7 (IC₅₀ = 7.1, 63 and 943 µM, |
Secondary target | SET7 |
Purity | ≥95% by HPLC |
Physicochemical Information | |
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Cell permeable | Y |
Dimensions |
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Safety Information according to GHS |
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Product Usage Statements |
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Packaging Information | |
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Packaged under inert gas | Packaged under inert gas |
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Supplemental Information |
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Specifications |
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Global Trade Item Number | |
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Catalogue Number | GTIN |
217531-10MG | 04055977219388 |
Documentation
CARM1 Inhibitor - CAS 1020399-49-8 - Calbiochem SDS
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CARM1 Inhibitor - CAS 1020399-49-8 - Calbiochem Certificates of Analysis
Title | Lot Number |
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217531 |
References
Reference overview |
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Cheng, D., et al. 2011. J. Med. Chem. 54, 4928. |