Adenosine A2A Rec.Antagon. II, SCH-58261

Name: Adenosine A2A Rec.Antagon. II, SCH-58261
Brand: MM

Synonym(s):

2-(furan-2-yl)-7-phenethyl-7H-pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine, SCH58261, SCH 58261

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About This Item

Linear Formula:

C18H15N7O

CAS Number:

160098-96-4

NACRES:

NA.51

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Properties

form

(Off-white solid)

Quality Segment

100

solubility

soluble (100 mM in DMSO)

storage temp.

2-8°C

Description

General description

A highly potent and selective antagonist of adenosine A2A receptor (Ki = 600 pM). Does not affect the activity of other adenosine receptors in any significant manner (Ki = 287 nM; 5.0 µM, and > 10 µM for A1, A2B, and A3 receptors, respectively). Displays neuroprotective effects in cerebral ischaemia in rats, and shown to counteract Parkinsonian-like muscle rigidity in rats.

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