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Merck

539604

PKCη Pseudosubstrate Inhibitor, Myristoylated

The PKCη Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKCη. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.

Synonym(s):

PKCη Pseudosubstrate Inhibitor, Myristoylated, Myr-TRKRQRAMRRRVHQING-OH, Protein Kinase C η Pseudosubstrate Inhibitor, Myristoylated

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About This Item

Empirical Formula (Hill Notation):
C101H185N41O23S
Molecular Weight:
2373.88
NACRES:
NA.77
UNSPSC Code:
12352200
Assay:
≥95% (HPLC)
Form:
lyophilized solid
Quality level:
Storage condition:
OK to freeze, desiccated (hygroscopic)
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Quality Level

assay

≥95% (HPLC)

form

lyophilized solid

manufacturer/tradename

Calbiochem®

storage condition

OK to freeze, desiccated (hygroscopic)

solubility

water: 1 mg/mL

shipped in

ambient

storage temp.

−20°C

General description

A cell-permeable, reversible, substrate competitive, and pseudosubstrate inhibitor of the protein kinase Cη isozyme. Useful for studies of PKCη function in intact cells.

Biochem/physiol Actions

Product competes with ATP.
Reversible: yes
Cell permeable: yes
Primary Target
PKCν

Packaging

Yes

Physical form

Supplied as a trifluoroacetate salt.

Preparation Note

Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 6 months at -20°C.

Other Notes

Myr-Thr-Arg-Lys-Arg-Gln-Arg-Ala-Met-Arg-Arg-Arg-Val-His-Gln-Ile-Asn-Gly-OH
Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.

Legal Information

CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany

Disclaimer

Toxicity: Standard Handling (A)


Storage Class

11 - Combustible Solids

wgk

WGK 1

flash_point_f

Not applicable

flash_point_c

Not applicable



Certificates of Analysis (COA)

Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.

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