539636
PKCθ Pseudosubstrate Inhibitor, Myristoylated
The PKCθ Pseudosubstrate Inhibitor, Myristoylated controls the biological activity of PKCθ. This small molecule/inhibitor is primarily used for Phosphorylation & Dephosphorylation applications.
Synonym(s):
PKCθ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH2, Protein Kinase C θ Pseudosubstrate Inhibitor, Myristoylated, Myr-LHQRRGAIKQAKVHHVKC-NH2, Protein Kinase Cθ Pseudosubstrate Inhibitor, Myristoylated
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About This Item
Empirical Formula (Hill Notation):
C105H182N35O22S
Molecular Weight:
2318.85
NACRES:
NA.77
UNSPSC Code:
12352200
Assay:
≥95% (HPLC)
Form:
lyophilized solid
Quality level:
Storage condition:
OK to freeze, desiccated (hygroscopic)
Quality Level
assay
≥95% (HPLC)
form
lyophilized solid
manufacturer/tradename
Calbiochem®
storage condition
OK to freeze, desiccated (hygroscopic)
solubility
water: 2 mg/mL
shipped in
ambient
storage temp.
−20°C
General description
A cell-permeable, reversible, substrate competitive, myristoylated form of the inhibitor of protein kinase Cθ isozyme pseudosubstrate inhibitor (Cat. No. 539634).
Cell-permeable myristoylated protein kinase Cq pseudosubstrate sequence peptide (Cat. No. 539634). Useful for studies of PKCθ function in intact cells. Sold on the basis of peptide content.
Biochem/physiol Actions
Cell permeable: yes
Primary Target
protein kinase Cθ
protein kinase Cθ
Product competes with ATP.
Reversible: yes
Physical form
Supplied as a trifluoroacetate salt.
Preparation Note
Following reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for 6 months at -20°C.
Other Notes
Myr-Leu-His-Gln-Arg-Arg-Gly-Ala-Ile-Lys-Gln-Ala-Lys-Val-His-His-Val-Lys-Cys-NH₂
Osada, S., et al. 1992. Mol. Cell Biol.12, 3930.
Legal Information
CALBIOCHEM is a registered trademark of Merck KGaA, Darmstadt, Germany
Disclaimer
Toxicity: Standard Handling (A)
Storage Class
11 - Combustible Solids
wgk
WGK 1
flash_point_f
Not applicable
flash_point_c
Not applicable
Certificates of Analysis (COA)
Search for Certificates of Analysis (COA) by entering the products Lot/Batch Number. Lot and Batch Numbers can be found on a product’s label following the words ‘Lot’ or ‘Batch’.
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