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505897 (±)-PD 128907 Hydrochloride - CAS 112960-16-4 - Calbiochem

505897
  
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Áttekintés

Replacement Information

Kulcsspecifikációk táblázata

CAS #Empirical Formula
112960-16-4C₁₄H₁₉NO₃•HCl
Description
Overview

This product has been discontinued.



Selective dopamine D3 receptor agonist (Ki = 2.3 nM) with an 18-fold selectivity over long dopamine receptors (D2L) and exhibited only weak affinity for D4.2 receptors (Ki = 169 nM). Commonly used to reproduce cocaine′s discriminative stimulus effects and also in peripheral systemic studies of hypertension.

Catalogue Number505897
Brand Family Calbiochem®
SynonymsDopamine D₃ Receptor Agonist, PD 128,907, PD 128907, PD128907
References
ReferencesAchat-Mendes, c. et al. 2010. J. Pharmacol. Exp. Ther. 334, 556.
Zeng, C. et al. 2006. Circul. Res. 99, 494.
Pugsley, T. A. et al. 1995. J. Pharmacol. Exp. Ther. 275, 1355.
Product Information
CAS number112960-16-4
FormWhite powder
Hill FormulaC₁₄H₁₉NO₃•HCl
Chemical formulaC₁₄H₁₉NO₃•HCl
Structure formula ImageStructure formula Image
Quality LevelMQ100
Applications
Biological Information
Primary TargetD₃
Primary Target K<sub>i</sub>2.3 nM
Purity≥98% by HPLC
Physicochemical Information
Dimensions
Materials Information
Toxicological Information
Safety Information according to GHS
Safety Information
Product Usage Statements
Storage and Shipping Information
Ship Code Shipped at Ambient Temperature or with Blue Ice or with Dry Ice
Toxicity Standard Handling
Storage -20°C
Protect from Light Protect from light
Do not freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Packaging Information
Transport Information
Supplemental Information
Specifications
Global Trade Item Number
Katalógusszám GTIN
505897 0

Documentation

(±)-PD 128907 Hydrochloride - CAS 112960-16-4 - Calbiochem MSDS

Title

Safety Data Sheet (SDS) 

References

Hivatkozások áttekintése
Achat-Mendes, c. et al. 2010. J. Pharmacol. Exp. Ther. 334, 556.
Zeng, C. et al. 2006. Circul. Res. 99, 494.
Pugsley, T. A. et al. 1995. J. Pharmacol. Exp. Ther. 275, 1355.

Brochure

Title
New Products Flyer- Feb 2014 - Vol 1
Data Sheet

Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

Revision20-September-2013 JSW
SynonymsDopamine D₃ Receptor Agonist, PD 128,907, PD 128907, PD128907
DescriptionSelective dopamine D3 receptor agonist (Ki = 2.3 nM) with an 18-fold selectivity over long dopamine receptors (D2L) and exhibited only weak affinity for D4.2 receptors (Ki = 169 nM). Commonly used to reproduce cocaine′s discriminative stimulus effects and also in peripheral systemic studies of hypertension.
FormWhite powder
CAS number112960-16-4
Chemical formulaC₁₄H₁₉NO₃•HCl
Structure formulaStructure formula
Purity≥98% by HPLC
SolubilityH₂O (5 mg/ml)
Storage Protect from light
-20°C
Do Not Freeze Ok to freeze
Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
Toxicity Standard Handling
ReferencesAchat-Mendes, c. et al. 2010. J. Pharmacol. Exp. Ther. 334, 556.
Zeng, C. et al. 2006. Circul. Res. 99, 494.
Pugsley, T. A. et al. 1995. J. Pharmacol. Exp. Ther. 275, 1355.