Millipore Sigma Vibrant Logo

05-23-3831 BQ-123, Sodium Salt - CAS - Calbiochem

A highly potent, selective, and competitive ETA (endothelin) receptor antagonist (Ki = 40 nM for ETA versus Ki = 2.5 µM for ETB).

BQ-123, Sodium Salt - CAS - Calbiochem MSDS (material safety data sheet) or SDS, CoA and CoQ, dossiers, brochures and other available documents.
Primary Target: ETA (endothelin) receptor antagonist
05-23-3831
View Pricing & Availability

Overview

Replacement Information

Key Spec Table

Empirical Formula
C₃₁H₄₁N₆O₇ · Na

Pricing & Availability

Catalogue Number AvailabilityPackaging Qty/Pack Price Quantity
05-23-3831-1MG
Retrieving availability...
—
Fulfilment and delivery delayed Fulfilment and delivery delayed
In Stock 
Discontinued
Limited Quantities Available
Availability to be confirmed
    Remaining : Will advise
      Remaining : Will advise
      Will advise
      Contact Customer Service
      Contact Customer Service

      		 Plastic ampoule 1 mg
      Retrieving price...
      Price could not be retrieved
      Minimum Quantity is a multiple of
      Maximum Quantity is
      Upon Order Completion More Information
      You Saved ()
       
      —
      Request Pricing
      		 —
      05-23-3831-5MG
      Retrieving availability...
      —
      Fulfilment and delivery delayed Fulfilment and delivery delayed
      In Stock 
      Discontinued
      Limited Quantities Available
      Availability to be confirmed
        Remaining : Will advise
          Remaining : Will advise
          Will advise
          Contact Customer Service
          Contact Customer Service

          		 Plastic ampoule 5 mg
          Retrieving price...
          Price could not be retrieved
          Minimum Quantity is a multiple of
          Maximum Quantity is
          Upon Order Completion More Information
          You Saved ()
           
          —
          Request Pricing
          		 —
          Description
          OverviewA highly potent, selective, and competitive ETA (endothelin) receptor antagonist (Ki = 40 nM for ETA versus Ki = 2.5 μM for ETB).
          Catalogue Number05-23-3831
          Brand Family Calbiochem®
          References
          ReferencesNambi, P., et al. 1996. J. Pharmacol. Exp. Ther. 277, 1567.
          Bax, W.A., and Saxena, P.R. 1994. Trends Pharmacol. Sci. 15, 379.
          Ihara, M., et al. 1991. Biochem. Biophys. Res. Commun. 178, 132.
          Product Information
          ATP CompetitiveN
          FormWhite solid
          FormulationSupplied as a sodium salt. Sold on the basis of peptide content.
          Hill FormulaC₃₁H₄₁N₆O₇ · Na
          Chemical formulaC₃₁H₄₁N₆O₇ · Na
          Hygroscopic Hygroscopic
          ReversibleN
          Sold on the basis of peptide contentY
          Quality LevelMQ100
          Applications
          Biological Information
          Primary TargetETA (endothelin) receptor antagonist
          Primary Target K<sub>i</sub>40 nM for ETA versus 2.5 µM for ETB
          Purity≥95% by HPLC
          Physicochemical Information
          Cell permeableN
          Peptide ContentY
          Peptide SequenceCyclo(D-Asp-Pro-D-Val-Leu-D-Trp, Na)
          Dimensions
          Materials Information
          Toxicological Information
          Safety Information according to GHS
          Safety Information
          Product Usage Statements
          Storage and Shipping Information
          Ship Code Ambient Temperature Only
          Toxicity Standard Handling
          Storage -20°C
          Hygroscopic Hygroscopic
          Do not freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Packaging Information
          Transport Information
          Supplemental Information
          Specifications

          Documentation

          BQ-123, Sodium Salt - CAS - Calbiochem SDS

          Title

          Safety Data Sheet (SDS) 

          BQ-123, Sodium Salt - CAS - Calbiochem Certificates of Analysis

          TitleLot Number
          05-23-3831

          References

          Reference overview
          Nambi, P., et al. 1996. J. Pharmacol. Exp. Ther. 277, 1567.
          Bax, W.A., and Saxena, P.R. 1994. Trends Pharmacol. Sci. 15, 379.
          Ihara, M., et al. 1991. Biochem. Biophys. Res. Commun. 178, 132.
          Data Sheet

          Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

          Revision31-May-2011 JSW
          DescriptionA highly potent and selective ETA (endothelin) receptor antagonist (Ki = 40 nM for ETA versus 2.5 µM for ETB).
          FormWhite solid
          FormulationSupplied as a sodium salt. Sold on the basis of peptide content.
          Chemical formulaC₃₁H₄₁N₆O₇ · Na
          Peptide SequenceCyclo(D-Asp-Pro-D-Val-Leu-D-Trp, Na)
          Purity≥95% by HPLC
          SolubilityH₂O (1 mg/ml)
          Storage -20°C
          Hygroscopic
          Do Not Freeze Ok to freeze
          Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 3 months at -20°C.
          Toxicity Standard Handling
          ReferencesNambi, P., et al. 1996. J. Pharmacol. Exp. Ther. 277, 1567.
          Bax, W.A., and Saxena, P.R. 1994. Trends Pharmacol. Sci. 15, 379.
          Ihara, M., et al. 1991. Biochem. Biophys. Res. Commun. 178, 132.