370654 PKG Inhibitor - Calbiochem

370654
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Overview

Replacement Information

Key Spec Table

Empirical Formula
C₃₈H₇₄N₁₈O₁₀

Pricing & Availability

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370654-1MGCN
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      Plastic ampoule 1 mg
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      Description
      OverviewA more specific, reversible, and substrate competitive inhibitor of protein kinase G (Ki = 86 µM) relative to protein kinase A (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35).
      Catalogue Number370654
      Brand Family Calbiochem®
      SynonymsProtein Kinase G Inhibitor, RKRARKE
      References
      ReferencesGlass, D.B., et al. 1983. Biochem. J. 213, 159.
      Product Information
      ATP CompetitiveN
      FormLyophilized
      Hill FormulaC₃₈H₇₄N₁₈O₁₀
      Chemical formulaC₃₈H₇₄N₁₈O₁₀
      Hygroscopic Hygroscopic
      ReversibleY
      Sold on the basis of peptide contentY
      Quality LevelMQ100
      Applications
      Biological Information
      Primary TargetPKG
      Primary Target K<sub>i</sub>86 µM against protein kinase G
      Purity≥95% by HPLC
      Physicochemical Information
      Cell permeableN
      Peptide ContentY
      Peptide SequenceH-Arg-Lys-Arg-Ala-Arg-Lys-Glu-OH
      Dimensions
      Materials Information
      Toxicological Information
      Safety Information according to GHS
      Safety Information
      Product Usage Statements
      Storage and Shipping Information
      Ship Code Ambient Temperature Only
      Toxicity Standard Handling
      Storage -20°C
      Hygroscopic Hygroscopic
      Do not freeze Ok to freeze
      Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 2 months at -20°C.
      Packaging Information
      Transport Information
      Supplemental Information
      Specifications

      Documentation

      PKG Inhibitor - Calbiochem Certificates of Analysis

      TitleLot Number
      370654

      References

      Reference overview
      Glass, D.B., et al. 1983. Biochem. J. 213, 159.
      Data Sheet

      Note that this data sheet is not lot-specific and is representative of the current specifications for this product. Please consult the vial label and the certificate of analysis for information on specific lots. Also note that shipping conditions may differ from storage conditions.

      Revision11-January-2010 RFH
      SynonymsProtein Kinase G Inhibitor, RKRARKE
      DescriptionA specific, reversible, and substrate competitive inhibitor of PKG (Ki = 86 µM) relative to PKA (Ki = 550 µM). Sequence corresponds to a non-phosphorylatable analog (Ser32 to Ala32) of histone H2B (amino acids 29-35).
      FormLyophilized
      Chemical formulaC₃₈H₇₄N₁₈O₁₀
      Peptide SequenceH-Arg-Lys-Arg-Ala-Arg-Lys-Glu-OH
      Purity≥95% by HPLC
      SolubilityH₂O (1 mg/ml)
      Storage -20°C
      Hygroscopic
      Do Not Freeze Ok to freeze
      Special InstructionsFollowing reconstitution, aliquot and freeze (-20°C). Stock solutions are stable for up to 2 months at -20°C.
      Toxicity Standard Handling
      ReferencesGlass, D.B., et al. 1983. Biochem. J. 213, 159.