Saltar al contenido
Merck

CHRM2

cholinergic receptor, muscarinic 2

Sinónimos:
HM2
Especie:
ID UniProtKB:
ID del gen:
  • Human(1129) Summary: The muscarinic cholinergic receptors belong to a larger family of G protein-coupled receptors. The functional diversity of these receptors is defined by the binding of acetylcholine to these receptors and includes cellular responses such as adenylate cyclase inhibition, phosphoinositide degeneration, and potassium channel mediation. Muscarinic receptors influence many effects of acetylcholine in the central and peripheral nervous system. The muscarinic cholinergic receptor 2 is involved in mediation of bradycardia and a decrease in cardiac contractility. Multiple alternatively spliced transcript variants have been described for this gene. [provided by RefSeq, Jul 2008]
  • Mouse(243764) cholinergic receptor, muscarinic 2, cardiac
  • Rat(81645) cholinergic receptor, muscarinic 2
  • Domestic Rabbit(100342878) cholinergic receptor, muscarinic 2
  • naked mole-rat(101714286) cholinergic receptor, muscarinic 2
  • chicken(418126) cholinergic receptor, muscarinic 2
  • domestic guinea pig(100715343) cholinergic receptor, muscarinic 2
  • dog(403858) cholinergic receptor, muscarinic 2
  • cow(522170) cholinergic receptor, muscarinic 2
  • domestic cat(101099790) cholinergic receptor, muscarinic 2
  • sheep(101102897) cholinergic receptor, muscarinic 2
  • sheep(100628317) cholinergic receptor, muscarinic 2

Custom & Knockdown Gene Products

  • siRNA

    Shop predesigned siRNA that are designed using the proprietary Rosetta Inpharmatics algorithm.

  • shRNA

    Shop the largest, most validated shRNA collection and build your own clone sets.

  • Custom Gene Products

    We offer a comprehensive portfolio of DNA oligos, RNA oligos and predesigned primers.

Small Molecule - Agonist

Product Number
Descripción
Especie
Pilocarpine hydrochloride, ≥99% (titration), powder,
Especie
human
Acetyl-β-methylcholine chloride, ≥98% (TLC), powder,
Especie
human
Pilocarpine nitrate salt, ≥98% (HPLC),
Especie
human
Oxotremorine M, solid,
Especie
human
(±)-Muscarine chloride hydrate, ≥98% (HPLC),
Especie
human

Small Molecule - Antagonist

Product Number
Descripción
Especie
Methoctramine hydrate, ≥97% (NMR), solid,
Especie
human
Darifenacin hydrobromide, ≥98% (HPLC),
Especie
human
Oxybutynin chloride, United States Pharmacopeia (USP) Reference Standard,
Especie
human
Oxybutynin hydrochloride, European Pharmacopoeia (EP) Reference Standard,
Especie
human
Darifenacin hydrobromide, United States Pharmacopeia (USP) Reference Standard,
Especie
human

Antibodies

Product Number
Descripción
Reactividad de especies
Aplicación
Anti-Muscarinic Acetylcholine Receptor m2 Antibody, clone M2-2-B3, clone M2-2-B3, Chemicon®, from rat,
Reactividad de especies
human, mammals, monkey, rat
Aplicación
immunocytochemistry
immunohistochemistry

immunoprecipitation (IP)
Anti-Muscarinic Acetylcholine Receptor M2 Antibody, Chemicon®, from rabbit,
Reactividad de especies
human
Aplicación
immunohistochemistry
Monoclonal Anti-CHRM2 antibody produced in mouse, clone 4B5, purified immunoglobulin, buffered aqueous solution,
Reactividad de especies
human
Aplicación
ELISA
western blot
Anti-CHRM2 antibody produced in mouse, purified immunoglobulin, buffered aqueous solution,
Reactividad de especies
human
Aplicación
western blot
Anti-Muscarinic AChR M2 (ACM2) Antibody, clone 3T5W8, Rabbit Monoclonal, ,
Reactividad de especies
human, rat
Aplicación
immunohistochemistry
western blot

Small Molecule - Inhibitor

Product Number
Descripción
Especie
(+)-Pentazocine, solid,
Especie
rat, human
Amitriptyline hydrochloride, ≥98% (TLC), powder,
Especie
human
Doxepin hydrochloride, ~85% E-isomer basis, ≥98% (GC), 15% Z-isomer basis, powder,
Especie
human
Haloperidol, powder,
Especie
human, rat
Harmaline, ≥95%,
Especie
human, rat

Small Molecule - Ligand

Product Number
Descripción
Especie
Aminobenztropine, solid,
Especie
human

Proteins

Product Number
Descripción
Especie
ChemiSCREEN Membrane Preparation Recombinant Human M2 Muscarinic Acetylcholine Receptor, Human M2 GPCR membrane prepation for Radioligand binding Assays.,
Especie
human

esiRNA

Product Number
Descripción
Especie
MISSION® esiRNA, targeting human CHRM2,
Especie
human