344152
FPT Inhibitor II
(E,E)-2-[2-Oxo-2-[[(3,7,11-trimethyl-2,6,10-dodecatrienyl)oxy]amino]ethyl]phosphonic Acid, 2Na
Untuk pertanyaan umum, silakan hubungi Layanan Pelanggan kami:
Merck KGaA
Frankfurter Str. 250
64293 Darmstadt
Germany
Telefon: +49 6151 72-0
Faks: +49 6151 72 2000
31 May 2012
memuat
A cell permeable potent and selective inhibitor of farnesyltransferase (FTase; IC50 = 75 nM). Also inhibits Ras farnesylation in whole cells by ~90% at 25-250 µM. Resistant to cleavage by phosphorylation.
| Informasi produk | |||
|---|---|---|---|
| Form | White solid | ||
| Primary Target | FTase | ||
| Primary Target IC50 | 75 nM | ||
| Hygrocopic | Ya | ||
| Cell permeable | Ya | ||
| Purity | ≥95% by TLC | ||
| Formulasi kimia | C17H28NO5P • 2Na • 3H2O | ||
| Simpan dan kirim informasi | |||
|---|---|---|---|
| Penyimpanan | -20°C | ||
| Ship |
Ambient Temperature Only
Standard Handling |
||
